Browsing BIOQBM - Artículos by Author "Lucio Ortega, Héctor Elessar de"
Now showing items 1-15 of 15
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Comparison of hydrocarbon-and lactam-bridged cyclic peptides as dimerization inhibitors of Leishmania infantum trypanothione reductase
Sánchez Murcia, Pedro Alejandro; Ruiz Santaquiteria, Marta; Toro Londoño, Miguel Ángel; Lucio Ortega, Héctor Elessar de; Jiménez , María Ángeles; [et al.] (2015-06-19) -
Efficient dimerization disruption of Leishmania infantum trypanothione reductase by triazole-phenyl-thiazoles
Revuelto Pérez, Alejandro; Lucio Ortega, Héctor Elessar de; García Soriano, Juan Carlos; Sánchez Murcia, Pedro Alejandro; Gago Badenas, Federico; [et al.] (2021-05-04) -
First example of peptides targeting the dimer interface of Leishmania infantum trypanothione reductase with potent in vitro antileishmanial activity
Ruiz Santaquiteria, Marta; Sánchez Murcia, Pedro Alejandro; Toro Londoño, Miguel Ángel; Lucio Ortega, Héctor Elessar de; Gutiérrez Viñas, Kilian Jesús; [et al.] (2017-07-28) -
A functional BH3 domain in an aquaporin from Leishmania infantum
Genes Robles, Carlos Mario; Lucio Ortega, Héctor Elessar de; Manuel González, Víctor; Sánchez Murcia, Pedro Alejandro; Rico , Eva; [et al.] (2016-07-04) -
Identification of 1,2,3-triazolium salt-based inhibitors of Leishmania infantum trypanothione disulfide reductase with enhanced antileishmanial potency in cellulo and increased selectivity
Lucio Ortega, Héctor Elessar de; Revuelto Pérez, Alejandro; Carriles Linares, Alejandra Ángela; De Castro De La Osa, Sonia; García González, Sonia; [et al.] (2022-10-29) -
Identification of L. infantum trypanothione synthetase inhibitors with leishmanicidal activity from a (non-biased) in-house chemical library
Alcón Calderón, María de las Mercedes; Lucio Ortega, Héctor Elessar de; García Soriano, Juan Carlos; Revuelto Pérez, Alejandro; De Castro De La Osa, Sonia; [et al.] (2022-08-18) -
Identification of NEK3 and MOK as novel targets for lithium
Bravo , Ana; Lucio Ortega, Héctor Elessar de; Sánchez Murcia, Pedro Alejandro; Jiménez Ruiz, Antonio; Petrone , Paula M.; [et al.] (2019-02-12) -
Improved proteolytic stability and potent activity against Leishmania infantum trypanothione reductase of alfa/beta-peptide foldamers conjugated to cell-penetrating peptides
Lucio Ortega, Héctor Elessar de; Gamo , Ana María; Ruiz Santaquiteria, Marta; De Castro , Sonia; Sánchez Murcia, Pedro Alejandro; [et al.] (2017-11-10) -
Next generation of selenocyanate and diselenides with upgraded leishmanicidal activity
Henríquez Figuereo, Andreina; Alcón Calderón, María de las Mercedes; Moreno Amatria, Esther; Sanmartín Grijalba, Carmen; Espuelas Millán, María Socorro; [et al.] (2023-05-24) -
Pro-death activity of a BH3 domain in an aquaporin from the protozoan parasite Leishmania
Genes Robles, Carlos Mario; Lucio Ortega, Héctor Elessar de; Sánchez Murcia, Pedro Alejandro; Gago Badenas, Federico; Jiménez Ruiz, Antonio (2016-07-28) -
Pseudoirreversible slow-binding inhibition of trypanothione reductase by a protein-protein interaction disruptor
Lucio Ortega, Héctor Elessar de; Toro Londoño, Miguel Ángel; Camarasa Rius, María José; Velázquez Díaz, Sonsoles; Gago Badenas, Federico; [et al.] (2020-10-02) -
Pyrrolopyrimidine vs Imidazole-Phenyl-Thiazole Scaffolds in Nonpeptidic Dimerization Inhibitors of Leishmania infantum Trypanothione Reductase
Revuelto , Alejandro; Ruiz Santaquiteria, Marta; Lucio Ortega, Héctor Elessar de; Gamo , Ana; Carriles Linares, Alejandra Ángela; [et al.] (2019-04-15) -
Small Molecule-Peptide Conjugates as Dimerization Inhibitors of Leishmania infantum Trypanothione Disulfide Reductase
Revuelto Pérez, Alejandro; López Martín, Isabel; Lucio Ortega, Héctor Elessar de; García Soriano, Juan Carlos; Zanda , Nicola; [et al.] (2021-07-17) -
Synthesis and Leishmanicidal Activity of Novel Urea, Thiourea, and Selenourea Derivatives of Diselenides
Díaz Hernando, Marta; Lucio Ortega, Héctor Elessar de; Moreno Amatria, Esther; Espuelas Millán, María Socorro; Aydillo Miguel, Carlos; [et al.] (2019-04-25) -
Trypanothione reductase inhibition and anti-leishmanial activity of all-hydrocarbon stapled alfa-helical peptides with improved proteolytic stability
Ruiz Santaquiteria, Marta; De Castro , Sonia; Toro, Miguel A.; Lucio Ortega, Héctor Elessar de; Gutiérrez Viñas, Kilian Jesús; [et al.] (2018-04-10)