Browsing by Author "Camarasa Rius, María José"
Now showing items 1-12 of 12
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Comparison of hydrocarbon-and lactam-bridged cyclic peptides as dimerization inhibitors of Leishmania infantum trypanothione reductase
Sánchez Murcia, Pedro Alejandro; Ruiz Santaquiteria, Marta; Toro Londoño, Miguel Ángel; Lucio Ortega, Héctor Elessar de; Jiménez , María Ángeles; [et al.] (2015-06-19) -
Dimerization inhibitors of HIV-1 reverse transcriptase, protease and integrase: A single mode of inhibition for the three HIV enzymes?
Camarasa Rius, María José; Velázquez Díaz, Sonsoles; San Félix García, Ana; Pérez Pérez, María Jesús; Gago Badenas, Federico (2006) -
Efficient dimerization disruption of Leishmania infantum trypanothione reductase by triazole-phenyl-thiazoles
Revuelto Pérez, Alejandro; Lucio Ortega, Héctor Elessar de; García Soriano, Juan Carlos; Sánchez Murcia, Pedro Alejandro; Gago Badenas, Federico; [et al.] (2021-05-04) -
Identification of 1,2,3-triazolium salt-based inhibitors of Leishmania infantum trypanothione disulfide reductase with enhanced antileishmanial potency in cellulo and increased selectivity
Lucio Ortega, Héctor Elessar de; Revuelto Pérez, Alejandro; Carriles Linares, Alejandra Ángela; De Castro De La Osa, Sonia; García González, Sonia; [et al.] (2022-10-29) -
Identification of aspartic acid-203 in human thymidine phosphorylase as an important residue for both catalysis and non-competitive inhibition by the small molecule "crystallization chaperone" 5'-O-tritylinosine (KIN59)
Bronckaers, A.; Aguado, L.; Negri Martínez, Ana; Camarasa Rius, María José; Balzarini, Jan; [et al.] (2009) -
Identification of L. infantum trypanothione synthetase inhibitors with leishmanicidal activity from a (non-biased) in-house chemical library
Alcón Calderón, María de las Mercedes; Lucio Ortega, Héctor Elessar de; García Soriano, Juan Carlos; Revuelto Pérez, Alejandro; De Castro De La Osa, Sonia; [et al.] (2022-08-18) -
Improved proteolytic stability and potent activity against Leishmania infantum trypanothione reductase of alfa/beta-peptide foldamers conjugated to cell-penetrating peptides
Lucio Ortega, Héctor Elessar de; Gamo , Ana María; Ruiz Santaquiteria, Marta; De Castro , Sonia; Sánchez Murcia, Pedro Alejandro; [et al.] (2017-11-10) -
The N137 and P140 amino acids in the p51 and the P95 amino acid in the p66 subunit of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase are instrumental to maintain catalytic activity and to design new classes of anti-HIV-1 drugs
Auwerx, Joeri; Nieuwenhove, Joke Van; Rodríguez Barrios, Fátima; Castro, Sonia de; Velázquez Díaz, Sonsoles; [et al.] (2005) -
Pseudoirreversible slow-binding inhibition of trypanothione reductase by a protein-protein interaction disruptor
Lucio Ortega, Héctor Elessar de; Toro Londoño, Miguel Ángel; Camarasa Rius, María José; Velázquez Díaz, Sonsoles; Gago Badenas, Federico; [et al.] (2020-10-02) -
Small Molecule-Peptide Conjugates as Dimerization Inhibitors of Leishmania infantum Trypanothione Disulfide Reductase
Revuelto Pérez, Alejandro; López Martín, Isabel; Lucio Ortega, Héctor Elessar de; García Soriano, Juan Carlos; Zanda , Nicola; [et al.] (2021-07-17) -
Trypanothione reductase inhibition and anti-leishmanial activity of all-hydrocarbon stapled alfa-helical peptides with improved proteolytic stability
Ruiz Santaquiteria, Marta; De Castro , Sonia; Toro, Miguel A.; Lucio Ortega, Héctor Elessar de; Gutiérrez Viñas, Kilian Jesús; [et al.] (2018-04-10) -
TSAO compounds: The comprehensive story of a unique family of HIV-1 specific inhibitors of reverse transcriptase
Camarasa Rius, María José; San Félix García, Ana; Velázquez Díaz, Sonsoles; Pérez Pérez, María Jesús; Gago Badenas, Federico; [et al.] (2004)